ClC(OCC)=O.[CH2:7]([O:9][C:10]([NH:12][CH2:13][C:14]([OH:16])=O)=[O:11])[CH3:8].C(N(CC)CC)C.[NH:24]([C:26]1[N:27]=[N:28][C:29]([C:33]2[CH:38]=[CH:37][CH:36]=[CH:35][CH:34]=2)=[C:30]([CH3:32])[N:31]=1)[NH2:25]>C(Cl)Cl.C(Cl)(Cl)Cl>[CH2:7]([O:9][C:10]([NH:12][CH2:13][C:14]([NH:25][NH:24][C:26]1[N:27]=[N:28][C:29]([C:33]2[CH:34]=[CH:35][CH:36]=[CH:37][CH:38]=2)=[C:30]([CH3:32])[N:31]=1)=[O:16])=[O:11])[CH3:8]A solution of ethyl chloroformate (3.689 g) in methylene chloride (10 ml) was added dropwise to a stirred solution of N-ethoxycarbonylglycine (4.998 g) and triethylamine (3.434 g) in methylene chloride (60 ml) under cooling in 5 minutes, and the stirring was continued for 5 minutes under cooling. To the solution of the mixed anhydride was added a solution of 3-hydrazino-5-methyl-6-phenyl-1,2,4-triazine (3.417 g) in chloroform (40 ml) and reacted in a similar manner to that of Example 17-(1). The reaction mixture was washed with water, dried over magnesium sulfate, and evaporated under reduced pressure. The residue was dissolved in ethanol (50 ml) and a solution of sodium hydroxide (1.6 g) in water (10 ml) was added dropwise to the solution with stirring under ice cooling in 5 minutes. After stirring for 30 minutes at room temperature, the solution was evaporated, and the residue was dissolved in a small amount of water. The solution was salted out and extracted with ethyl acetate. The extract was washed with a saturated aqueous solution of sodium chloride, dried over magnesium sulfate, and evaporated. The residue was dissolved in chloroform containing a small amount of ethanol and the solution was chromatographed on silica gel (50 g). The eluent with a mixture of chloroform and ethanol (30:1) gave a colorless solid of 3-[2-(N-ethoxycarbonylglycyl)hydrazino]-5-methyl-6-phenyl-1,2,4-triazine (1.872 g).
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