Phenylboronic Acid → 6-Phenylpyridin-3-amine
Reaction equation
Br[C:2]1[N:7]=[CH:6][C:5]([NH2:8])=[CH:4][CH:3]=1.[C:9]1(B(O)O)[CH:14]=[CH:13][CH:12]=[CH:11][CH:10]=1>>[C:9]1([C:2]2[N:7]=[CH:6][C:5]([NH2:8])=[CH:4][CH:3]=2)[CH:14]=[CH:13][CH:12]=[CH:11][CH:10]=1Participants
3
Procedure
Obtained (71% yield) following the procedure described in Intermediate 39, starting with 6-bromopyridin-3-amine and phenylboronic acid.
Workup
- customObtained (71% yield)
Sources & evidence
- ORD record
- ord-1c7968cc267e4180bc4bdd30cf07bfa8
- Source dataset
- uspto-grants-2013_09
- Patent number
- US08536165B2
Reaction notes
Loading…