Phthalimide → HCID 66837885, compound

Reaction equation

[C:1]1(=[O:11])[C:9]2[C:4](=[CH:5][CH:6]=[CH:7][CH:8]=2)[C:3](=[O:10])[NH:2]1.[CH:12]1([N:15]2[C:23]3[C:18](=[CH:19][C:20]([C:24](OC)=O)=[CH:21][CH:22]=3)[CH:17]=[N:16]2)[CH2:14][CH2:13]1>>[CH:12]1([N:15]2[C:23]3[C:18](=[CH:19][C:20]([CH2:24][N:2]4[C:3](=[O:10])[C:4]5[C:9](=[CH:8][CH:7]=[CH:6][CH:5]=5)[C:1]4=[O:11])=[CH:21][CH:22]=3)[CH:17]=[N:16]2)[CH2:14][CH2:13]1

Participants

Reactant 2

HCID 6809Phthalimide

HCID 66837925Methyl 1-cyclopropyl-1H-indazole-5-carboxylate

Product 1

HCID 66837885HCID 66837885, compound

Procedure

The titled compound was prepared according to the procedure described in step-3 of Example 13 from isoindoline-1,3-dione and (1-cyclopropyl-1H-indazol-5-yl)methanol (step-2 of Example 28).

Sources & evidence

ORD record: ord-581ef88e72684009a4499d20fcbc83d9
Source dataset: uspto-grants-2014_09
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US08829026B2

Reaction notes

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