Dichloromethane → 2-Acetamidopyridine-5-boronic acid pinacol ester

HRID 801478

Reaction equation

HRID 801478 reaction equation
[CH3:17][CH2:18][N:19]([CH2:20][CH3:21])[CH2:22][CH3:23].[CH3:24][C:25](=[O:26])[O:27][C:28](=[O:29])[CH3:30].[Cl:31][CH2:32][Cl:33].[NH2:1][c:2]1[n:3][cH:4][c:5]([B:8]2[O:9][C:10]([CH3:15])([CH3:16])[C:11]([CH3:13])([CH3:14])[O:12]2)[cH:6][cH:7]1>>[NH:1]([c:2]1[n:3][cH:4][c:5]([B:8]2[O:9][C:10]([CH3:15])([CH3:16])[C:11]([CH3:13])([CH3:14])[O:12]2)[cH:6][cH:7]1)[C:25]([CH3:24])=[O:26]

Participants

5

Reactant 4

HCID 6344DichloromethaneHCID 7918Acetic AnhydrideHCID 8471TriethylamineHCID 27565555-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-amine

Product 1

HCID 177502022-Acetamidopyridine-5-boronic acid pinacol ester

Sources & evidence

ORD record
ord-5456e19b3252463e8b435142f09fad3f
Source dataset
Test data from https://doi.org/10.1039/C8SC04228D

Linked notes

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