反応式
[F:1][C:2]1[CH:3]=[C:4]2[C:8](=[CH:9][CH:10]=1)[NH:7][CH:6]=[C:5]2[CH:11]=[O:12].[CH2:13](OC(C1NC2C(C=1)=CC=CC=2)=O)[CH3:14]>>[CH2:13]([N:7]1[C:8]2[C:4](=[CH:3][C:2]([F:1])=[CH:10][CH:9]=2)[C:5]([CH:11]=[O:12])=[CH:6]1)[CH3:14]参加物
3
実験手順
According to the procedure of Preparation 9 (a), except substituting 5-fluoro-1H-indole-3-carboxaldehyde (0.41 g, 2.5 mmole) for the ethylindole-2-carboxylate, the title compound (0.20 g, 57%) was prepared as a viscous oil: MS (ES) m/e 191 (M+H)+.
出典と根拠
- ORDレコード
- ord-22b7264a9a4a4c3cb7ea6fc693fa027d
- 出典データセット
- uspto-grants-2010_06
- 特許番号
- US07741339B2
関連ノート
読み込み中…