反応式
[F:1][C:2]1[CH:3]=[C:4]2[C:8](=[CH:9][CH:10]=1)[N:7]([CH3:11])[C:6]([C:12]([O:14]CC)=O)=[CH:5]2.[CH3:17][N:18]1C2C(=CC=CC=2)C=C1C(OCC)=O>>[CH3:17][NH:18][C:12]([C:6]1[N:7]([CH3:11])[C:8]2[C:4]([CH:5]=1)=[CH:3][C:2]([F:1])=[CH:10][CH:9]=2)=[O:14]参加物
3
実験手順
According to the procedure of Preparation 1(b), except substituting ethyl 5-fluoro-1-methyl-1H-indole-2-carboxylate for the ethyl 1-methyl-1H-indole-2-carboxylate, the title compound (2.1 g, 68%) was prepared as a white solid: MS (ES) m/e 207 (M+H)+.
出典と根拠
- ORDレコード
- ord-5937838202174a5190a842483394e586
- 出典データセット
- uspto-grants-2009_07
- 特許番号
- US07557125B2
関連ノート
読み込み中…