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(Naphthalen-2-yl)boronic acid → 3-(Naphthalen-2-yl)-1-trityl-1H-pyrazolo[4,3-b]pyridine
関与物質
| 役割 | 名称 | HCID | 仕込み量 |
|---|---|---|---|
| 反応物 | (Naphthalen-2-yl)boronic acid | HCID 2734375 | — |
| 反応物 | 3-Iodo-1-trityl-1H-pyrazolo[4,3-b]pyridine | HCID 68932363 | — |
| 生成物 | 3-(Naphthalen-2-yl)-1-trityl-1H-pyrazolo[4,3-b]pyridine | HCID 68932700 | 28.7% |
反応手順
By treating 731 mg of 3-iodo-1-trityl-1H-pyrazolo[4,3-b]pyridine obtained by Example 418 and 340 mg of 2-naphthalene boronic acid in the manner as described in Production example 194, 210 mg of the title compound was obtained as a colorless powder.
情報源と証拠
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| 特許番号 | US07429609B2 |
| 出典データセット | uspto-grants-2008_09 |
| ORD ID | ord-fe5376172d2748c08c3fccc8b5ac8ca6 |
| 出典メモ | uspto-grants-2008_09 |