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HRID 57616作成日：2026年10月26日

(4-(Morpholin-4-yl)phenyl)boronic acid → Tert-butyl 3-hydroxy-5-((7-(4-morpholinophenyl)pyrido[4,3-b]pyrazin-5-ylamino)methyl)piperidine-1-carboxylate

https://huagongshe.com/reaction/57616

反応式

関与物質

役割名称HCID仕込み量
反応物(4-(Morpholin-4-yl)phenyl)boronic acidHCID 2795359—
反応物Tert-butyl 3-((7-chloropyrido[4,3-b]pyrazin-5-ylamino)methyl)-5-hydroxypiperidine-1-carboxylateHCID 86717368—
生成物Tert-butyl 3-hydroxy-5-((7-(4-morpholinophenyl)pyrido[4,3-b]pyrazin-5-ylamino)methyl)piperidine-1-carboxylateHCID 71113447—

反応手順

The title compound was prepared according to the procedures of Compound 1 (B) using tert-butyl 3-((7-chloropyrido[4,3-b]pyrazin-5-ylamino)methyl)-5-hydroxypiperidine-1-carboxylate and 4-morpholinophenylboronic acid. MS (m/z): 521 (M+H)+.

情報源と証拠

DOI10.6084/m9.figshare.5104873.v1
特許番号US09434726B2
出典データセットuspto-grants-2016_09
ORD IDord-e599baed4a414dda88e024d000d4e251
出典メモuspto-grants-2016_09