Benzocaine → HCID 178468129, 화합물

HRID 1722087노트

반응식

HRID 1722087 반응식
[CH2:1]([P:3](Cl)(=[O:11])[O:4][C:5]1[CH:10]=CC=CC=1)[CH3:2].[CH2:13]([O:15][C:16](=[O:20])[CH2:17][CH2:18][NH2:19])[CH3:14].[CH2:21](OC(=O)CCN)[C:22]1[CH:27]=[CH:26][CH:25]=[CH:24][CH:23]=1.[CH2:34]([O:36]C(=O)C1C=CC(N)=CC=1)[CH3:35].C([O:53]C(=O)C1C=CC(N)=CC=1)C1C=CC=CC=1>>[CH2:13]([O:15][C:16](=[O:20])[CH2:17][CH2:18][NH:19][C:10](=[O:53])[C@@H:5]([O:4][PH:3]([CH2:1][CH2:2][O:36][CH2:34][CH3:35])=[O:11])[CH2:21][C:22]1[CH:23]=[CH:24][CH:25]=[CH:26][CH:27]=1)[CH3:14]

참가 물질

6

반응물 5

HCID 2337BenzocaineHCID 98488Benzyl p-aminobenzoateHCID 419889Ethyl 3-aminopropanoateHCID 1116164Benzyl 3-aminopropanoateHCID 20030345Phenyl ethyl-phosphonochloridate

생성물 1

HCID 178468129HCID 178468129, 화합물

실험 절차

Use the same procedure substituting ethyl ethylphosphonochloridate with the appropriate aralkyl ethylphosphonochloridate or phenyl ethyl-phosphonochloridate and when necessary substituting N-(S)-phenyllactoyl) β-alanine ethyl ester with N-(S)-phenyllactoyl) β-alanine benzyl ester, N-(S)-phenyllactoyl) p-aminobenzoic acid ethyl ester or N-(S)-phenyllactoyl) p-aminobenzoic acid benzyl ester and synthesize compounds 3, 6, 8, 11, 13, 16, 18, 21, 23, 31 or 33.

출처 및 근거

ORD 기록
ord-d08d63928f134b8fb3e63bb2f30dbfb5
출처 데이터셋
uspto-grants-1989_08
특허 번호
US04853476

반응 노트

불러오는 중…