4-(((tert-Butoxycarbonyl)amino)methyl)benzoic acid → tert-Butyl (4-{[((1R,2S)-2-{[(3aR,4R,9bR)-4-(methoxymethyl)-2,3,3a,4,5,9b-hexahydro-1H-pyrrolo[3,2-c]quinolin-1-yl]carbonyl}cyclohexyl)amino]carbonyl}benzyl)carbamate

Beteiligte Stoffe

Rolle	Name	HCID	Einwaage
Edukt	4-(((tert-Butoxycarbonyl)amino)methyl)benzoic acid	HCID 853605	—
Edukt	(1R,2S)-2-{[(3aR,4R,9bR)-4-(methoxymethyl)-2,3,3a,4,5,9b-hexahydro-1H-pyrrolo[3,2-c]quinolin-1-yl]carbonyl}cyclohexaneamine dihydrochloride	HCID 67150533	—
Produkt	tert-Butyl (4-{[((1R,2S)-2-{[(3aR,4R,9bR)-4-(methoxymethyl)-2,3,3a,4,5,9b-hexahydro-1H-pyrrolo[3,2-c]quinolin-1-yl]carbonyl}cyclohexyl)amino]carbonyl}benzyl)carbamate	HCID 57846897	—

Reaktionsschritte

In the same manner as in Reference Example 19 and using 4-{[(tert-butoxycarbonyl)amino]methyl}benzoic acid and (1R,2S)-2-{[(3aR,4R,9bR)-4-(methoxymethyl)-2,3,3a,4,5,9b-hexahydro-1H-pyrrolo[3,2-c]quinolin-1-yl]carbonyl}cyclohexaneamine dihydrochloride, the title compound was synthesized.

Herkunft & Nachweise

DOI	10.6084/m9.figshare.5104873.v1
Patentnummer	US07973163B2
Quelldatensatz	uspto-grants-2011_07
ORD ID	ord-67edc4d982154a1eacf1370a6322c4cf
Quellennotiz	uspto-grants-2011_07