HRID1043592

反应详情

EQUATION

反应方程式

HRID 1043592 的结构方程式

PROCEDURE

实验过程

2-(4-((2-Chloro-4-morpholinopyrido[3,2-d]pyrimidin-6-yl)methyl)piperazin-1-yl)-2-methylpropanamide from Example 121 (115 mg) was reacted with 2-aminopyridine-5-boronic acid, pinacol ester via General Procedure A to yield 8.5 mg 124 following reverse phase HPLC purification. MS (Q1) 492.3 (M)+

WORKUP

后处理

  1. customto yield
  2. custom8.5 mg 124 following reverse phase HPLC purification