HuagongsheHuagongshe Chemistry Print Report · For research reference only
1-Amino-3-(4-chloro-phenyl)-propan-2-one hydrochloride → 3-benzyloxy-7-morpholin-4-yl-4-oxo-4H-pyrido[1,2-a]pyrimidine-2-carboxylic acid [3-(4-chloro-phenyl)-2-oxo-propyl]-amide
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 1-Amino-3-(4-chloro-phenyl)-propan-2-one hydrochloride | HCID 13290676 | — |
| Reactant | 3-benzyloxy-7-morpholin-4-yl-4-oxo-4H-pyrido[1,2-a]pyrimidine-2-carboxylic acid | HCID 57494573 | — |
| Product | 3-benzyloxy-7-morpholin-4-yl-4-oxo-4H-pyrido[1,2-a]pyrimidine-2-carboxylic acid [3-(4-chloro-phenyl)-2-oxo-propyl]-amide | HCID 66953269 | — |
Reaction Steps
Adapted the procedure of example 2 using 3-benzyloxy-7-morpholin-4-yl-4-oxo-4H-pyrido[1,2-a]pyrimidine-2-carboxylic acid and 1-amino-3-(4-chloro-phenyl)-propan-2-one hydrochloride (AU2007001980) as starting material
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08563562B2 |
| Source dataset | uspto-grants-2013_10 |
| ORD ID | ord-8d2ea4fe0f094cecbf0b22129a415c00 |
| Source note | uspto-grants-2013_10 |