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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1061004Generated: November 1, 2026

4-(Diethylboranyl)pyridine → 1-[2-tert-Butoxycarbonyl-4-(pyridin-4-yl)benzoyl]-4-[(6-chloronaphthalen-2-yl)sulfonyl]piperazine hydrochloride

https://huagongshe.com/reaction/1061004

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-(Diethylboranyl)pyridineHCID 13318871—
Reactant1-[4-Bromo-2-(tert-butoxycarbonyl)benzoyl]-4-[(6-chloronaphthalen-2-yl)sulfonyl]piperazineHCID 22709864—
Product1-[2-tert-Butoxycarbonyl-4-(pyridin-4-yl)benzoyl]-4-[(6-chloronaphthalen-2-yl)sulfonyl]piperazine hydrochlorideHCID 22710746—

Reaction Steps

In a similar manner to Referential Example 7 except for the use of 1-[4-bromo-2-(tert-butoxycarbonyl)benzoyl]-4-[(6-chloronaphthalen-2-yl)sulfonyl]piperazine and diethyl(4-pyridyl)borane as the raw materials, the reaction was conducted, whereby the title compound was obtained.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS06525042B1
Source datasetuspto-grants-2003_02
ORD IDord-31417add813c4a56a6eb35184e0572fd
Source noteuspto-grants-2003_02