[2-Chloro-4-(trifluoromethyl)phenyl]boronic acid → HCID 11642285, compound

Participants

Reaction Steps

The title compound is prepared by following a procedure analogous to Example 113, Step 1, using N-{2-[(2-dimethylamino-ethyl)-methyl-amino]-benzothiazol-6-yl}-4-iodo-benzamide (0.10 g, 0.21 mmol) and 2-chloro-4-trifluoromethyl-phenyl boronic acid (0.056 g, 0.25 mmol) to afford 0.045 g (40%). LC/MS, Retention time=5.34 min; (m/z): calcd for C26H24ClF3N4OS: 533.0; found: 533.0.

Provenance & Evidence