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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1244389Generated: November 2, 2026

2-Methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenol → HCID 136122457, compound

https://huagongshe.com/reaction/1244389

Reaction equation

Participants

RoleNameHCIDCharge
Reactant2-Methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenolHCID 2734650—
Reactant6-Chloro-N-[(1R)-1-(4-methylphenyl)ethyl]pyrazin-2-amineHCID 58717110—
ProductHCID 136122457HCID 1361224576.5%

Reaction Steps

In a procedure analogous to Example 2, reaction of 6-chloro-N-[(1R)-1-(4-methylphenyl)ethyl]pyrazin-2-amine (56.8 mg, 0.229 mmol) and 2-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenol 63 mg, 0.25 mmol) furnished the product (5 mg, 6%).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07122550B2
Source datasetuspto-grants-2006_10
ORD IDord-2380ab7bc2264ceaa04cee7f3f21bec1
Source noteuspto-grants-2006_10