2-Bromobenzaldehyde → HCID 21904933, compound

Participants

Reaction Steps

In analogy to example 262.2, (RS)-N-(4-cyano-benzyl)-2-[2,6-difluoro-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-phenyl]-2-ethoxy-acetamide (example 262.1) was reacted with 2-bromobenzaldehyde to give (RS)-N-(4-cyano-benzyl)-2-(3,5-difluoro-2′-formyl-biphenyl-4-yl)-2-ethoxy-acetamide. Off-white solid. MS 435.0 ([M+H]+)

Provenance & Evidence