3-Amino-3-methyloxetane → HCID 57378671, compound

Participants

Reaction Steps

As described for example 3b, 4-{4-[5-(4-fluoro-phenyl)-3-methyl-3H-[1,2,3]triazol-4-yl]-imidazol-1-yl}-benzoic acid (75 mg, 0.21 mmol) was converted, using 3-methyl-3-oxetanamine instead of isopropylamine, to the title compound (57 mg, 64%) which was obtained as a white solid after trituration from ethyl acetate. MS: m/e=433.4 [M+H]+.

Provenance & Evidence