2-(Methylamino)-1-[4-(pyrrolidin-1-yl)phenyl]ethan-1-ol → 7-Oxo-4,5,6,7-tetrahydro-benzo[b]thiophene-3-sulfonic acid [2-hydroxy-2-(4-pyrrolidine-1-yl-phenyl)-ethyl]-methyl-amide

Participants

Reaction Steps

From 2-methylamino-1-(4-pyrrolidine-1-yl-phenyl)-ethanol (the compound of Preparation Example 19) (63 mg) and 7-oxo-4,5,6,7-tetrahydro-benzo[b]thiophene-3-sulfonyl chloride (the compound of Preparation Example 7) (70 mg), the title compound (35 mg) was obtained as a colorless amorphous substance, in the same way as Preparation Example 41.

Provenance & Evidence