HuagongsheHuagongshe Chemistry Print Report · For research reference only
2-(S),5-Diamino-pentanoic acid [3-phenyl-1-(R)-(quinolin-3-ylcarbamoyl)-propyl]-amide mono-methanesulfonate → L-ornithyl-(3,4,5-trifluoro)-D-phenylalanine Quinoline-3-amide Mesylate
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 2-(S),5-Diamino-pentanoic acid [3-phenyl-1-(R)-(quinolin-3-ylcarbamoyl)-propyl]-amide mono-methanesulfonate | HCID 11663539 | — |
| Reactant | bis-Boc-L-ornithyl-(3,4,5-trifluoro)-D-Phenylalanine Quinoline-3-amide | HCID 86602424 | — |
| Product | L-ornithyl-(3,4,5-trifluoro)-D-phenylalanine Quinoline-3-amide Mesylate | HCID 86602422 | — |
Reaction Steps
NaNd-bis-Boc-L-ornithyl-(3,4,5-trifluoro)-D-Phenylalanine Quinoline-3-amide was converted into mono-mesylate salt of the tile product according to the procedure described for compound 3 to give the title product (0.15 g) as off white solid.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07893020B2 |
| Source dataset | uspto-grants-2011_02 |
| ORD ID | ord-90f72fe61c33407ca33111411e4b7e16 |
| Source note | uspto-grants-2011_02 |