4-Cyclopropylbenzoic acid → HCID 178523638, compound

Participants

Reaction Steps

The title compound, light yellow solid (85 mg, 72%), MS (ISP) m/z=471.4 [(M+H)+], mp 199° C., was prepared in accordance with the general method of example 1 from trans-4-[2-(4-benzofuran-3-yl-piperidin-1-yl)-ethyl]-cyclohexylamine dihydrochloride (intermediate A) (100 mg, 0.25 mmol) and 4-cyclopropyl-benzoic acid.

Provenance & Evidence