2-{5-Methyl-2-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)phenyl]-oxazol-4-yl}-ethanol → 2-{2-[4-(6-Ethanesulfonyl-pyridin-3-yl)-phenyl]-5-methyl-oxazol-4-yl}-ethanol

Participants

Reaction Steps

The titled compound is prepared substantially in accordance with the procedure of Intermediate 9 using 2-{5-Methyl-2-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)phenyl]-oxazol-4-yl}-ethanol (See Intermediate 3) and 2-Ethanesulfonyl-5-iodo-pyridine (See Intermediate 22). MS (m/e) 373.3 (M+1)

Provenance & Evidence