HuagongsheHuagongshe Chemistry Print Report · For research reference only
4-(Ethylsulphonyl)benzeneboronic acid → 2-(4'-Ethanesulfonyl-biphenyl-4-yl)-5-methyl-4-(2-pyrrolidin-1-yl-ethyl)-oxazole
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 4-(Ethylsulphonyl)benzeneboronic acid | HCID 2773420 | — |
| Reactant | 2-(4-Bromo-phenyl)-5-methyl-4-(2-pyrrolidin-1-yl-ethyl)-oxazole | HCID 11681546 | — |
| Product | 2-(4'-Ethanesulfonyl-biphenyl-4-yl)-5-methyl-4-(2-pyrrolidin-1-yl-ethyl)-oxazole | HCID 11582638 | — |
Reaction Steps
The title compound is prepared in a mamler substantially analogous to Example 35 starting from 4-Ethylsulfonylbenzene boronic acid and 2-(4-Bromo-phenyl)-5-methyl-4-(2-pyrrolidin-1-yl-ethyl)-oxazole. MS (m/e): 425.1 (M+1)
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07666871B2 |
| Source dataset | uspto-grants-2010_02 |
| ORD ID | ord-bdcf9a77df06423a9b852100acf9523f |
| Source note | uspto-grants-2010_02 |