4-(Trifluoromethoxy)phenylboronic acid → HCID 58951459, compound

Participants

Reaction Steps

The title compound is prepared in a manner substantially analogous to example 133 starting from 4-triflouromethoxy phenyl boronic acid (295 mg, 1.43 mmol) and 2-(4-Bromo-phenyl)-5-methyl-4-[2-((R)-2-methyl-pyrrolidin-1-yl)-ethyl]-oxazole (100 mg, 0.287 mmol) to give 63 mg (51%). MS (m/e) 431.2 (M+1)

Provenance & Evidence