HuagongsheHuagongshe Chemistry Print Report · For research reference only
5-N-Boc-amino-1H-indole → 1-(2-((1-(5-ethylpyrazin-2-yl)piperidin-4-yl)oxy)thiazol-4-yl)-1H-indol-5-amine
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 5-N-Boc-amino-1H-indole | HCID 11458923 | — |
| Reactant | HCID 67608573 | HCID 67608573 | — |
| Product | 1-(2-((1-(5-ethylpyrazin-2-yl)piperidin-4-yl)oxy)thiazol-4-yl)-1H-indol-5-amine | HCID 67617301 | — |
Reaction Steps
The title compound was prepared by following the similar procedure as described in Intermediate-27 using 4-bromo-2-((1-(5-ethylpyrazin-2-yl)piperidin-4-yl)oxy)thiazole and tert-butyl-1H-indol-5-ylcarbamate (0.092 g, 40%); MS: 421.2 (M+1).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09000175B2 |
| Source dataset | uspto-grants-2015_04 |
| ORD ID | ord-c142fde7752b4c1c81c003bfe4df6f56 |
| Source note | uspto-grants-2015_04 |