5-Amino-2-chlorophenol → HCID 68491242, compound

Participants

Reaction Conditions

Reaction Steps

Following the general procedure for the synthesis of 2-R-5-(heteroaryl-2-ylamino)phenol, 4-amino-2-chloropyrimidine (70 mg, 0.5 mmol) and 5-amino-2-chlorophenol (78 mg, 0.5 mmol) in 10% aqueous EtOH (2 mL) was heated at 90° C. for 18 h. The title compound was obtained in 47% yield a (60 mg) and used for the next step without additional purification.

Provenance & Evidence