HuagongsheHuagongshe Chemie-Druckbericht · Nur für Forschungszwecke
[5-(Trifluoromethyl)pyridin-3-yl]boronic acid → 4-(tert-Butyl)-2-((tert-butylamino)methyl)-6-(5-(trifluoromethyl)pyridin-3-yl)phenol
Beteiligte Stoffe
| Rolle | Name | HCID | Einwaage |
|---|---|---|---|
| Edukt | [5-(Trifluoromethyl)pyridin-3-yl]boronic acid | HCID 45158900 | — |
| Edukt | 8-bromo-3,6-di-tert-butyl-3,4-dihydro-2H-benzo[e][1,3]oxazine | HCID 86718559 | — |
| Produkt | 4-(tert-Butyl)-2-((tert-butylamino)methyl)-6-(5-(trifluoromethyl)pyridin-3-yl)phenol | HCID 86718565 | — |
Reaktionsschritte
The title compound was prepared as a white solid using the procedure described in Example 1 from 8-bromo-3,6-di-tert-butyl-3,4-dihydro-2H-benzo[e][1,3]oxazine (Intermediate 1) and 3-(trifluoromethyl)pyridine-5-boronic acid [Intermediate 2].
Herkunft & Nachweise
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patentnummer | US09409893B2 |
| Quelldatensatz | uspto-grants-2016_08 |
| ORD ID | ord-9d22387ac6d14a1c80e8e8a5ba7b162a |
| Quellennotiz | uspto-grants-2016_08 |