1-Methylindole → 1-methyl-3-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole

HRID 1490643Notes

Reaction equation

HRID 1490643 reaction equation
Cn1ccc2ccccc21>CC1(C)OBOC1(C)C.F[B-](F)(F)c1ccccc1[NH+]1CCCCC1>Cn1cc(B2OC(C)(C)C(C)(C)O2)c2ccccc21

Participants

4

Reactant 1

HCID 117811-Methylindole

Product 1

HCID 230580031-methyl-3-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indoleYield 80%

Reagents, catalysts & solvents 2

HCID 27347684,4,5,5-Tetramethyl[1,3,2]dioxaborolaneReagentHCID 140919606Trifluoro-(2-piperidin-1-ium-1-ylphenyl)boranuideCatalyst

Conditions

Temperature
80 °C

Sources & evidence

ORD record
ord-f27a7cb8b7d449c5b118b81874db47a9
Source dataset
Borylation dataset from Roche

Reaction notes

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