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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1490643Generated: October 30, 2026

1-Methylindole → 1-methyl-3-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole

https://huagongshe.com/reaction/1490643

Reaction equation

Participants

RoleNameHCIDCharge
Reactant1-MethylindoleHCID 11781—
Reagent4,4,5,5-Tetramethyl[1,3,2]dioxaborolaneHCID 2734768—
CatalystTrifluoro-(2-piperidin-1-ium-1-ylphenyl)boranuideHCID 140919606—
Product1-methyl-3-(tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indoleHCID 2305800380%

Reaction Conditions

Temperature80 °C

Provenance & Evidence

DOI10.1021/jacs.7b08143
Source datasetBorylation dataset from Roche
ORD IDord-f27a7cb8b7d449c5b118b81874db47a9
Source noteBorylation dataset from Roche