Triethylamine → HCID 49848904, compound

Participants

Reaction Steps

The same reaction as in the method described in Example 2 was performed using the tert-butyl 4-({5-methyl-6-[5-(methylsulfonyl)indolin-1-yl]pyrimidin-4-yl}oxy)piperidine-1-carboxylate (208 mg, 0.426 mmol) produced in Example 26 and, instead of triethylamine, diisopropylethylamine (380 μL, 2.13 mmol) to obtain the title compound as white foam (177 mg, yield: 88%).

Provenance & Evidence