Methanesulfonyl chloride → HCID 86677488, compound

Participants

Reaction Steps

The product was obtained starting from 2-(2-(2-ethylpyridin-4-yl)-5-methylthiazol-4-yl)ethanol (200 mg, 805 μmol, prepared as described in WO 2003/037327) and methanesulfonyl chloride (111 mg, 75.3 μL, 966 μmol) according to the method described in example 46, step 1 as yellow oil (226 mg, 692 μmol, 86%) which was used without further purification for the next step.

Provenance & Evidence