HCID 20080599, compound → HCID 58201665, compound

Participants

Reaction Steps

The title compound was prepared in analogy to Example 5 starting from 1-iodo-2-methanesulfonyl-benzene (commercially available) and 3-{[phenyl-(3-phenyl propynoyl)-amino]-methyl}-benzoic acid methyl ester. 1H NMR (300 Hz, CDCl3): δppm 1.89 (s, 1.5H), 2.50 (s, 1.5H), 3.90 (s, 3H), 4.98 (dd, 2H), 5.98 (dd, 1H), 6.65-6.68 (m, 2H), 7.07 (m, 1H), 7.35-7.58 (m, 8H), 7.61 (t, 1H), 7.78 (t, 1H), 7.99 (d, 1H), 8.02 (d, 1H), 8.20 (d, 1H).

Provenance & Evidence