HuagongsheHuagongshe Chemistry Print Report · For research reference only
3-chloro-4-fluoro-N-hydroxy-benzenecarboximidamide → HCID 58002409, compound
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 3-chloro-4-fluoro-N-hydroxy-benzenecarboximidamide | HCID 4411739 | — |
| Reactant | 5-(4-Ethylphenyl)-1-(morpholin-4-ylcarbonyl)piperidine-3-carboxylic acid | HCID 58002225 | — |
| Product | HCID 58002409 | HCID 58002409 | — |
Reaction Steps
69 mg (0.20 mmol) of 5-(4-ethylphenyl)-1-(morpholin-4-ylcarbonyl)piperidine-3-carboxylic acid (Example 38A) and 41 mg (0.22 mmol, 1.1 eq.) of 3-chloro-4-fluoro-N′-hydroxybenzenecarboximidamide were reacted according to the General Method 1. Yield: 51 mg (51% of theory)
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08119663B2 |
| Source dataset | uspto-grants-2012_02 |
| ORD ID | ord-2ee1a524658f46d4b121392c08549756 |
| Source note | uspto-grants-2012_02 |