1-Aminopiperidine → HCID 59568393, compound

Participants

Reaction Steps

As described for example 26d, 5-(3-butyl-5-methyl-isoxazol-4-ylmethoxy)-2H-pyrazole-3-carboxylic acid methyl ester (218 mg, 0.74 mmol) was converted, using 1-aminopiperidine instead of 4-aminotetrahydropyran, to the title compound (228 mg, 85%) which was obtained as a colorless oil. MS: m/e=362.2 [M+H]+.

Provenance & Evidence