1-Propanol, 3-amino-2,2-dimethyl- → HCID 59568390, compound

Participants

Reaction Steps

As described for example 55, 5-[3-(4-fluoro-phenyl)-5-methyl-isoxazol-4-ylmethoxy]-2-methyl-2H-pyrazole-3-carboxylic acid (100 mg, 0.3 mmol) was converted, using 3-amino-2,2-dimethyl-1-propanol instead of 2-amino-2-methyl-1-propanol, to the title compound (88 mg, 70%) which was obtained as a white solid. MS: m/e=417.2 [M+H]+.

Provenance & Evidence