3-Amino-3-methyloxetane → HCID 59568402, compound

Participants

Reaction Steps

As described for example 160c, 1-methyl-3-((5-methyl-3-(pyridin-2-yl)isoxazol-4-yl)methylamino)-1H-pyrazole-5-carboxylic acid (80 mg, 255 μmol) was converted, using 3-methyl-3-oxetanamine instead of isopropylamine, to the title compound (68 mg, 70%) which was obtained as a white solid. MS: m/e=383.3 [M+H]+.

Provenance & Evidence