Cyclopropylamine → HCID 59568394, compound

Participants

Reaction Steps

As described for example 163c, 3-((3-(5-fluoropyridin-2-yl)-5-methylisoxazol-4-yl)methylamino)-1-methyl-1H-pyrazole-5-carboxylic acid (92 mg, 0.28 mol) was converted, using cyclopropylamine instead of isopropylamine, to the title compound (78 mg, 76%) which was obtained as a white solid. MS: m/e=371.3 [M+H]+.

Provenance & Evidence