2-Amino-6-(trifluoromethyl)pyridine → HCID 178488331, compound

Participants

Reaction Steps

The title compound (28 mg, 12%), light brown foam, MS (ISP): m/e=457.3 (M+H+), was prepared in accordance with the general method of Example 35 from rac-(6-bromo-4H-benzo[d][1,3]oxazin-2-yl)-(4-methoxy-2,3-dihydro-benzofuran-3-yl)-amine (Example 54) (188 mg, 0.5 mmol) and commercially available 2-amino-6-trifluoromethyl-pyridine (162 mg, 1.0 mmol).

Provenance & Evidence