Morpholine → HCID 178521232, compound

Participants

Reaction Steps

Prepared from 2-chloro-N-[2-(2-phenoxy-ethylamino)-4H-benzo[d][1,3]oxazin-6-yl]-acetamide (Example 122, step A) (180 mg, 0.50 mmol; HPLC 1.096 min) and morpholine (0.87 ml, 10 mmol) according to the procedure described for Example 3 step B. Obtained the title compound as a white solid (206 mg, 100%; HPLC 0.588 min), MS (ISP) m/e=411.2 [(M+H)+].

Provenance & Evidence