Phenylboronic Acid → HCID 66748461, compound

HRID 1747899Notes

Reaction equation

HRID 1747899 reaction equation
Br.Br[C:3]1[O:7][C:6]([C:8]2[C:9]([NH2:14])=[N:10][CH:11]=[CH:12][CH:13]=2)=[CH:5][CH:4]=1.[C:15]1(B(O)O)[CH:20]=[CH:19][CH:18]=[CH:17][CH:16]=1>>[C:15]1([C:3]2[O:7][C:6]([C:8]3[C:9]([NH2:14])=[N:10][CH:11]=[CH:12][CH:13]=3)=[CH:5][CH:4]=2)[CH:20]=[CH:19][CH:18]=[CH:17][CH:16]=1

Participants

3

Reactant 2

HCID 66827Phenylboronic AcidHCID 66747810HCID 66747810, compound

Product 1

HCID 66748461HCID 66748461, compound

Procedure

In the same manner as in Example 14, step A, the title compound (1.19 g) was obtained as a yellow solid from 3-(5-bromofuran-2-yl)pyridin-2-amine hydrobromide and phenylboronic acid.

Sources & evidence

ORD record
ord-f6a8da737390456fb61739f459d7704f
Source dataset
uspto-grants-2015_10
Patent number
US09150591B2

Reaction notes

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