Hydrogen iodide → HCID 51355566, compound

HRID 1751996Notes

Reaction equation

HRID 1751996 reaction equation
[C:1]([NH:4][C:5]1[CH:6]=[C:7](B(O)O)[CH:8]=[CH:9][CH:10]=1)(=[O:3])[CH3:2].Cl[C:15]1[CH:20]=[C:19](Cl)[N:18]=[CH:17][N:16]=1.[IH:22]>>[I:22][C:15]1[CH:20]=[C:19]([C:7]2[CH:8]=[CH:9][CH:10]=[C:5]([NH:4][C:1](=[O:3])[CH3:2])[CH:6]=2)[N:18]=[CH:17][N:16]=1

Participants

4

Reactant 3

HCID 24841Hydrogen iodideHCID 709434,6-DichloropyrimidineHCID 157274(3-Acetamidophenyl)boronic acid

Product 1

HCID 51355566HCID 51355566, compound

Procedure

The compound was prepared according to Example 1 using 3-acetylaminophenylboronic acid and 4,6-dichloropyrimidine. The resultant chloro compound was converted to iodo with hydroiodic acid as described in the general procedure.

Workup

  1. customThe compound was prepared

Sources & evidence

ORD record
ord-345532daa681436b85c8ec627f7de015
Source dataset
uspto-grants-2015_10
Patent number
US09162987B2

Reaction notes

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