Hydrogen iodide → HCID 51355845, compound

HRID 1752005Notes

Reaction equation

HRID 1752005 reaction equation
N[NH:2][C:3]([C:5]1[CH:10]=[CH:9][C:8](B(O)O)=[CH:7][CH:6]=1)=[O:4].Cl[C:15]1[CH:20]=[C:19](Cl)[N:18]=[CH:17][N:16]=1.[IH:22]>>[I:22][C:15]1[CH:20]=[C:19]([C:8]2[CH:9]=[CH:10][C:5]([C:3]([NH2:2])=[O:4])=[CH:6][CH:7]=2)[N:18]=[CH:17][N:16]=1

Participants

4

Reactant 3

HCID 24841Hydrogen iodideHCID 709434,6-DichloropyrimidineHCID 44119530[4-(Hydrazinecarbonyl)phenyl]boronic acid

Product 1

HCID 51355845HCID 51355845, compound

Procedure

The compound was prepared according to Example 1 using 4-aminocarbamoylphenylboronic acid and 4,6-dichloropyrimidine. The resultant chloro compound was converted to iodo with hydroiodic acid as described in the general procedure.

Workup

  1. customThe compound was prepared

Sources & evidence

ORD record
ord-84bfeeda80b942088ba3b769a9acb2db
Source dataset
uspto-grants-2015_10
Patent number
US09162987B2

Reaction notes

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