HuagongsheHuagongshe Chemistry Print Report · For research reference only
2-(2,4-Difluorobenzyloxy)-5-bromophenylboronic acid → 3-{2-[5-Bromo-2-(2,4-difluorobenzyloxy)phenyl]cyclopent-1-enyl}-5-aminobenzoic Acid Methyl Ester
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 2-(2,4-Difluorobenzyloxy)-5-bromophenylboronic acid | HCID 21112904 | — |
| Reactant | 3-Amino-5-(2-bromocyclopent-1-enyl)benzoic acid methyl ester | HCID 58887669 | — |
| Product | 3-{2-[5-Bromo-2-(2,4-difluorobenzyloxy)phenyl]cyclopent-1-enyl}-5-aminobenzoic Acid Methyl Ester | HCID 69507836 | — |
Reaction Steps
Prepared by general procedure 3 but using 3-amino-5-(2-bromocyclopent-1-enyl)benzoic acid methyl ester instead of 3-(2-bromocyclopent-1-enyl)benzoic acid ethyl ester and 2-(2,4-difluorobenzyloxy)-5-bromophenylboronic acid instead of 5-chloro-2-methoxyphenylboronic acid.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07232821B2 |
| Source dataset | uspto-grants-2007_06 |
| ORD ID | ord-6f3ad823a1db4898b516db0b82c68e16 |
| Source note | uspto-grants-2007_06 |