Pyrazole → HCID 86681300, compound

HRID 1778846Notes

Reaction equation

HRID 1778846 reaction equation
CN(C)[C:3]1[CH:4]=[C:5]([CH2:9]O)[CH:6]=[CH:7][CH:8]=1.[NH:12]1[CH:16]=[CH:15][CH:14]=[N:13]1.[CH3:17]C1(C)C(C)(C)OB(C2C=NNC=2)O1>>[CH3:17][C:5]1([CH2:9][N:12]2[CH:16]=[CH:15][CH:14]=[N:13]2)[CH2:4][CH2:3][CH2:8][CH2:7][CH2:6]1

Participants

4

Reactant 3

HCID 1048PyrazoleHCID 90133m-(Dimethylamino)benzyl alcoholHCID 27740104-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole

Product 1

HCID 86681300HCID 86681300, compound

Procedure

The title compound was prepared by substituting EXAMPLE 82A for (3-(dimethylamino)phenyl)methanol and 1H-pyrazole for 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole in EXAMPLE 34A.

Sources & evidence

ORD record
ord-c2d59eebca164fe3b2a62916fd167285
Source dataset
uspto-grants-2016_02
Patent number
US09266877B2

Reaction notes

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