HuagongsheHuagongshe Chemie-Druckbericht · Nur für Forschungszwecke
3-Cyclohexyl-2-[[1-cyclohexyl-2-(2-phenylquinoxalin-6-yl)benzimidazole-5-carbonyl]amino]propanoic acid → 2-[[1-Cyclohexyl-2-(2-phenylquinoxalin-6-yl)benzimidazole-5-carbonyl]amino]-3-phenyl-propanoic acid
Beteiligte Stoffe
| Rolle | Name | HCID | Einwaage |
|---|---|---|---|
| Edukt | 3-Cyclohexyl-2-[[1-cyclohexyl-2-(2-phenylquinoxalin-6-yl)benzimidazole-5-carbonyl]amino]propanoic acid | HCID 5276167 | — |
| Edukt | 9H-Fluoren-9-ylmethyl N-((1S)-1-formyl-2-phenylethyl)carbamate | HCID 10474375 | — |
| Produkt | 2-[[1-Cyclohexyl-2-(2-phenylquinoxalin-6-yl)benzimidazole-5-carbonyl]amino]-3-phenyl-propanoic acid | HCID 5276171 | 44% |
Reaktionsschritte
The general procedure described for Compound 242 was used with Fmoc-Phe Wang resin (167 mg, 0.6 mmol/g), producing 26 mg of the title compound (44% yield). MS: 594.24 (M−H+) HPLC Procedure A, retention time=14.58 min.
Herkunft & Nachweise
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patentnummer | US07511145B2 |
| Quelldatensatz | uspto-grants-2009_03 |
| ORD ID | ord-15200b5071cc425b84d0e423c16c6a4f |
| Quellennotiz | uspto-grants-2009_03 |