Piperidin-4-ol → HCID 5276193, compound

HRID 1788437Notes

Reaction equation

HRID 1788437 reaction equation
[Cl:1][C:2]1[CH:42]=[CH:41][C:5]([C:6]2[C:11]([C:12]3[CH:21]=[CH:20][C:19]4[C:14](=[CH:15][C:16]([F:40])=[C:17]([C:22]5[N:26]([CH:27]6[CH2:32][CH2:31][CH2:30][CH2:29][CH2:28]6)[C:25]6[CH:33]=[CH:34][C:35]([C:37](O)=[O:38])=[CH:36][C:24]=6[N:23]=5)[CH:18]=4)[N:13]=3)=[CH:10][CH:9]=[CH:8][CH:7]=2)=[CH:4][CH:3]=1.[OH:43][CH:44]1[CH2:49][CH2:48][NH:47][CH2:46][CH2:45]1>>[Cl:1][C:2]1[CH:42]=[CH:41][C:5]([C:6]2[C:11]([C:12]3[CH:21]=[CH:20][C:19]4[C:14](=[CH:15][C:16]([F:40])=[C:17]([C:22]5[N:26]([CH:27]6[CH2:32][CH2:31][CH2:30][CH2:29][CH2:28]6)[C:25]6[CH:33]=[CH:34][C:35]([C:37]([N:47]7[CH2:48][CH2:49][CH:44]([OH:43])[CH2:45][CH2:46]7)=[O:38])=[CH:36][C:24]=6[N:23]=5)[CH:18]=4)[N:13]=3)=[CH:10][CH:9]=[CH:8][CH:7]=2)=[CH:4][CH:3]=1

Participants

3

Reactant 2

HCID 79341Piperidin-4-olHCID 5276028HCID 5276028, compound

Product 1

HCID 5276193HCID 5276193, compound

Procedure

The title compound was synthesized from Compound 408 and 4-hydroxypiperidine using standard HBTU activation.

Sources & evidence

ORD record
ord-417b95c144e346c1a204a500c786e324
Source dataset
uspto-grants-2009_03
Patent number
US07511145B2

Reaction notes

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