1-(2-Pyrrolidin-1-YL-ethyl)-1H-indazol-6-ylamine → HCID 11430678, compound

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Reaction Steps

According to the procedure for Example 49, 1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-ylamine and 3-(5-p-tolyl-oxazol-2-yl)-propionic acid were processed to provide the title compound. MS (DCI/NH3) MS m/z 444 (M+H)+. 1H NMR (500 MHz, DMSO-d6) δ ppm 1.82 (m, 2 H), 1.98 (m, 2 H), 2.32 (s, 3 H), 2.93 (t, J=7.02 Hz, 2 H), 3.03 (m, 2 H), 3.15 (t, J=7.02 Hz, 2 H), 3.52 (m, 2 H), 3.69 (q, J=5.93 Hz, 2 H), 4.67 (t, J=6.24 Hz, 2 H), 7.10 (m, 1 H), 7.25 (m, 2 H), 7.47 (s, 1 H), 7.55 (m, 2 H), 7.71 (m, 1 H), 8.08 (s, 1 H), 8.31 (s, 1 H), 9.60 (br s, N H).

Provenance & Evidence