HCID 226349, compound → HCID 22036617, compound

Participants

Reaction Steps

According to the procedure for Example 49, 1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-ylamine and 3-(4-benzyloxy-3-methoxy-phenyl)-acrylic acid were processed to provide the title compound. MS (DCI/NH3) MS m/z 497 (M+H)+; 1H NMR (500 MHz, DMSO-d6) δ ppm 1.85 (m, 2 H), 2.01 (m, 2 H), 3.06 (m, 2 H), 3.55 (m, 2 H), 3.71 (m, 2H), 3.85 (s, 3 H), 4.71 (t, J=6.24 Hz, 2 H), 5.15 (s, 2 H), 6.79 (m, 1 H), 7.12 (m, 1 H), 7.18 (m, 2 H), 7.26 (m, 1 H), 7.35 (m, 1 H), 7.41 (m, 2 H), 7.46 (m, 2 H), 7.55 (m, 1 H), 7.74 (m, 1 H), 8.10 (s, 1 H), 8.41 (s, 1 H), 9.63 (br s, N H).

Provenance & Evidence