HuagongsheHuagongshe Chemistry Print Report · For research reference only
4-Morpholin-4-yl-4-oxo-2-benzylsulfonylmethyl-butyric acid → 4-Morpholin-4-yl-4-oxo-2-phenylmethanesulfonylmethyl-N-[(S)-1-(5-trifluoromethyl-1,2,4-oxadiazole-3-carbonyl)-propyl]-butyramide
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 4-Morpholin-4-yl-4-oxo-2-benzylsulfonylmethyl-butyric acid | HCID 22053987 | — |
| Reactant | (S)-2-amino-1-(5-trifluoromethyl-1,2,4-oxadiazol-3-yl)-butan-1-ol trifluoroacetate | HCID 86588340 | — |
| Product | 4-Morpholin-4-yl-4-oxo-2-phenylmethanesulfonylmethyl-N-[(S)-1-(5-trifluoromethyl-1,2,4-oxadiazole-3-carbonyl)-propyl]-butyramide | HCID 58619528 | — |
Reaction Steps
It is similarly prepared according to general procedure given for Example 2 above but using 4-Morpholin-4-yl-4-oxo-2-phenylmethanesulfonylmethyl-butyric acid and (S)-2-Amino-1-(5-trifluoromethyl-1,2,4-oxadiazol-3-yl)-butan-1-ol; compound with trifluoroacetic acid.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US07030116B2 |
| Source dataset | uspto-grants-2006_04 |
| ORD ID | ord-9d6d8e404f0e43df98e3d59576e9802c |
| Source note | uspto-grants-2006_04 |