2-(5''-Bromo-[2,2';4',3'']terpyridin-6'-yl)-propan-2-ol → 2-[5''-(1-Piperidin-4-yl-1H-pyrazol-4-yl)-[2,2';4',3'']terpyridin-6'-yl]-propan-2-ol

Participants

Role	Name	HCID	Charge
Reactant	2-(5''-Bromo-[2,2';4',3'']terpyridin-6'-yl)-propan-2-ol	HCID 68735197	—
Reactant	Methyl-[5''-(1-piperidin-4-yl-1H-pyrazol-4-yl)-[2,2';4',3'']terpyridin-6'-yl]-amine	HCID 68757252	—
Product	2-[5''-(1-Piperidin-4-yl-1H-pyrazol-4-yl)-[2,2';4',3'']terpyridin-6'-yl]-propan-2-ol	HCID 68761646	—

Reaction Steps

is prepared analogously to Methyl-[5″-(1-piperidin-4-yl-1H-pyrazol-4-yl)-[2,2′;4′,3″]terpyridin-6′-yl]-amine (Example 2.183) by replacing (5″-Bromo-[2,2′;4′,3″]terpyridin-6′-yl)-methyl-amine (Example 2.1; step 1) with 2-(5″-Bromo-[2,2′;4′,3″]terpyridin-6′-yl)-propan-2-ol (Example 2.80; step2)

Provenance & Evidence

DOI	10.6084/m9.figshare.5104873.v1
Patent number	US08343966B2
Source dataset	uspto-grants-2013_01
ORD ID	ord-bb132a1331bb4e80a75928e2123361ae
Source note	uspto-grants-2013_01