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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 1867845Generated: November 1, 2026

4-Bromo-2-fluorobenzoic acid → HCID 57980062, compound

https://huagongshe.com/reaction/1867845

Reaction equation

Participants

RoleNameHCIDCharge
Reactant4-Bromo-2-fluorobenzoic acidHCID 302681—
Reactant4-(Ethylsulphonyl)benzeneboronic acidHCID 2773420—
Reactant(R)-2-methyl-1-((S)-pyrrolidin-2-ylmethyl)pyrrolidineHCID 46911921—
ProductHCID 57980062HCID 57980062—

Reaction Steps

The title compound is prepared in a manner substantially analogous to Procedure A′, T′ and B′ starting from 4-bromo-2-fluoro-benzoic acid, 4-ethanesulfonylphenyl boronic acid and 2-(R)-Methyl-1-(2-(S)-pyrrolidinylmethyl)pyrrolidine. MS (M+H) 459.2

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07632857B2
Source datasetuspto-grants-2009_12
ORD IDord-6c0d3118343a4b929441f6bff0f8d7fd
Source noteuspto-grants-2009_12